Histaminski H1 receptor — разлика између измена

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== Reference ==
== Reference ==
{{Reflist|2}}
{{Reflist|2}}

== Literatura ==
{{refbegin | 2}}
{{PBB_Further_reading
| citations =
*{{cite journal | author=Mitsuchashi M, Payan DG |title=Molecular and cellular analysis of histamine H1 receptors on cultured smooth muscle cells. |journal=J. Cell. Biochem. |volume=40 |issue= 2 |pages= 183–92 |year= 1989 |pmid= 2670975 |doi= 10.1002/jcb.240400207 }}
*{{cite journal | author=Braman SS |title=Histamine receptors in the lung. |journal=N Engl Reg Allergy Proc |volume=8 |issue= 2 |pages= 116–20 |year= 1987 |pmid= 2886904 |doi=10.2500/108854187778994446 }}
*{{cite journal | author=Hill SJ, Ganellin CR, Timmerman H, ''et al.'' |title=International Union of Pharmacology. XIII. Classification of histamine receptors. |journal=Pharmacol. Rev. |volume=49 |issue= 3 |pages= 253–78 |year= 1997 |pmid= 9311023 |doi= }}
*{{cite journal | author=Holden CA, Chan SC, Norris S, Hanifin JM |title=Histamine induced elevation of cyclic AMP phosphodiesterase activity in human monocytes. |journal=Agents Actions |volume=22 |issue= 1–2 |pages= 36–42 |year= 1988 |pmid= 2891264 |doi=10.1007/BF01968814 }}
*{{cite journal | author=Moguilevsky N, Varsalona F, Noyer M, ''et al.'' |title=Stable expression of human H1-histamine-receptor cDNA in Chinese hamster ovary cells. Pharmacological characterisation of the protein, tissue distribution of messenger RNA and chromosomal localisation of the gene |journal=Eur. J. Biochem. |volume=224 |issue= 2 |pages= 489–95 |year= 1994 |pmid= 7925364 |doi=10.1111/j.1432-1033.1994.00489.x }}
*{{cite journal | author=Fukui H, Fujimoto K, Mizuguchi H, ''et al.'' |title=Molecular cloning of the human histamine H1 receptor gene |journal=Biochem. Biophys. Res. Commun. |volume=201 |issue= 2 |pages= 894–901 |year= 1994 |pmid= 8003029 |doi= 10.1006/bbrc.1994.1786 }}
*{{cite journal | author=Le Coniat M, Traiffort E, Ruat M, ''et al.'' |title=Chromosomal localization of the human histamine H1-receptor gene |journal=Hum. Genet. |volume=94 |issue= 2 |pages= 186–8 |year= 1994 |pmid= 8045566 |doi= }}
*{{cite journal | author=De Backer MD, Gommeren W, Moereels H, ''et al.'' |title=Genomic cloning, heterologous expression and pharmacological characterization of a human histamine H1 receptor |journal=Biochem. Biophys. Res. Commun. |volume=197 |issue= 3 |pages= 1601–8 |year= 1994 |pmid= 8280179 |doi=10.1006/bbrc.1993.2662 }}
*{{cite journal | author=Hishinuma S, Young JM |title=Characteristics of the binding of [3H]-mepyramine to intact human U373 MG astrocytoma cells: evidence for histamine-induced H1-receptor internalisation |journal=Br. J. Pharmacol. |volume=116 |issue= 6 |pages= 2715–23 |year= 1996 |pmid= 8590995 |doi= | pmc=1909113 }}
*{{cite journal | author=Max SI, Chowdhury BA, Fraser CM |title=Sequence analysis of the 5'-untranslated region of the human H1 histamine receptor-encoding gene |journal=Gene |volume=171 |issue= 2 |pages= 309–10 |year= 1996 |pmid= 8666296 |doi=10.1016/0378-1119(96)00036-4 }}
*{{cite journal | author=De Backer MD, Loonen I, Verhasselt P, ''et al.'' |title=Structure of the human histamine H1 receptor gene |journal=Biochem. J. |volume=335 |issue= 3|pages= 663–70 |year= 1998 |pmid= 9794809 |doi= | pmc=1219830 }}
*{{cite journal | author=Horváth BV, Szalai C, Mándi Y, ''et al.'' |title=Histamine and histamine-receptor antagonists modify gene expression and biosynthesis of interferon gamma in peripheral human blood mononuclear cells and in CD19-depleted cell subsets |journal=Immunol. Lett. |volume=70 |issue= 2 |pages= 95–9 |year= 1999 |pmid= 10569698 |doi=10.1016/S0165-2478(99)00126-1 }}
*{{cite journal | author=Wang KY, Arima N, Higuchi S, ''et al.'' |title=Switch of histamine receptor expression from H2 to H1 during differentiation of monocytes into macrophages |journal=FEBS Lett. |volume=473 |issue= 3 |pages= 345–8 |year= 2000 |pmid= 10818238 |doi=10.1016/S0014-5793(00)01560-X }}
*{{cite journal | author=Oda T, Morikawa N, Saito Y, ''et al.'' |title=Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes |journal=J. Biol. Chem. |volume=275 |issue= 47 |pages= 36781–6 |year= 2001 |pmid= 10973974 |doi= 10.1074/jbc.M006480200 }}
*{{cite journal | author=Brew OB, Sullivan MH |title=Localisation of mRNAs for diamine oxidase and histamine receptors H1 and H2, at the feto-maternal interface of human pregnancy |journal=Inflamm. Res. |volume=50 |issue= 9 |pages= 449–52 |year= 2002 |pmid= 11603849 |doi=10.1007/PL00000269 }}
*{{cite journal | author=Gutzmer R, Langer K, Lisewski M, ''et al.'' |title=Expression and function of histamine receptors 1 and 2 on human monocyte-derived dendritic cells |journal=J. Allergy Clin. Immunol. |volume=109 |issue= 3 |pages= 524–31 |year= 2002 |pmid= 11898002 |doi=10.1067/mai.2002.121944 }}
*{{cite journal | author=Idzko M, la Sala A, Ferrari D, ''et al.'' |title=Expression and function of histamine receptors in human monocyte-derived dendritic cells |journal=J. Allergy Clin. Immunol. |volume=109 |issue= 5 |pages= 839–46 |year= 2002 |pmid= 11994709 |doi=10.1067/mai.2002.124044 }}
}}
{{refend}}


== Vidi još ==
== Vidi još ==

Верзија на датум 9. мај 2012. у 17:54

Histamine receptor H1
Histaminski H1 receptor u kompleksu sa doksepinom (3RZE​)
Dostupne strukture
3RZE​
Identifikatori
Simboli HRH1; H1-R; hisH1
Vanjski ID OMIM: 600167 MGI: 107619 HomoloGene: 668 IUPHAR: H1 GeneCards: HRH1 Gene
Pregled RNK izražavanja
podaci
Ortolozi
Vrsta Čovek Miš
Entrez 3269 15465
Ensembl ENSG00000196639 ENSMUSG00000053004
UniProt P35367 P70174
RefSeq (mRNA) NM_000861.3 NM_001252642.1
RefSeq (protein) NP_000852.1 NP_001239571.1
Lokacija (UCSC) Chr 3:
11.18 - 11.31 Mb		 Chr 6:
114.35 - 114.43 Mb
PubMed pretraga [1] [2]

H1 receptor je histaminski receptor iz familije rodopsinu sličnih G protein spregnutih receptora. Ovaj receptor, koji aktivira biogeni amin histamin, je izražen širom tela, u glatkim mišićima, vaskularnim endotelnim ćelijama, u srcu, i u centralnom nervnom sistemu. H1 receptor je spregnut sa intracelularnim G proteinom (Gq) koji aktivira signalni put fosfolipaze C i fosfatidilinozitola (PIP2). Antihistamini koji deluju na ovaj receptor se koriste kao lekovi protiv alergije. Kristalna struktura receptora je određena.[1]

Reference

  1. ^ Tatsuro Shimamura, Mitsunori Shiroishi, Simone Weyand, Hirokazu Tsujimoto, Graeme Winter, Vsevolod Katritch, Ruben Abagyan, Vadim Cherezov, Wei Liu, Gye Won Han, Takuya Kobayashi, Raymond C. Stevens & So Iwata (2011). „Structure of the human histamine H1 receptor complex with doxepin”. Nature. 475 (7354): 65—70. PMID 21697825. doi:10.1038/nature10236.  Непознати параметар |month= игнорисан (помоћ)

Literatura

  • Mitsuchashi M, Payan DG (1989). „Molecular and cellular analysis of histamine H1 receptors on cultured smooth muscle cells.”. J. Cell. Biochem. 40 (2): 183—92. PMID 2670975. doi:10.1002/jcb.240400207. 
  • Braman SS (1987). „Histamine receptors in the lung.”. N Engl Reg Allergy Proc. 8 (2): 116—20. PMID 2886904. doi:10.2500/108854187778994446. 
  • Hill SJ, Ganellin CR, Timmerman H; et al. (1997). „International Union of Pharmacology. XIII. Classification of histamine receptors.”. Pharmacol. Rev. 49 (3): 253—78. PMID 9311023. 
  • Holden CA, Chan SC, Norris S, Hanifin JM (1988). „Histamine induced elevation of cyclic AMP phosphodiesterase activity in human monocytes.”. Agents Actions. 22 (1–2): 36—42. PMID 2891264. doi:10.1007/BF01968814. 
  • Moguilevsky N, Varsalona F, Noyer M; et al. (1994). „Stable expression of human H1-histamine-receptor cDNA in Chinese hamster ovary cells. Pharmacological characterisation of the protein, tissue distribution of messenger RNA and chromosomal localisation of the gene”. Eur. J. Biochem. 224 (2): 489—95. PMID 7925364. doi:10.1111/j.1432-1033.1994.00489.x. 
  • Fukui H, Fujimoto K, Mizuguchi H; et al. (1994). „Molecular cloning of the human histamine H1 receptor gene”. Biochem. Biophys. Res. Commun. 201 (2): 894—901. PMID 8003029. doi:10.1006/bbrc.1994.1786. 
  • Le Coniat M, Traiffort E, Ruat M; et al. (1994). „Chromosomal localization of the human histamine H1-receptor gene”. Hum. Genet. 94 (2): 186—8. PMID 8045566. 
  • De Backer MD, Gommeren W, Moereels H; et al. (1994). „Genomic cloning, heterologous expression and pharmacological characterization of a human histamine H1 receptor”. Biochem. Biophys. Res. Commun. 197 (3): 1601—8. PMID 8280179. doi:10.1006/bbrc.1993.2662. 
  • Hishinuma S, Young JM (1996). „Characteristics of the binding of [3H]-mepyramine to intact human U373 MG astrocytoma cells: evidence for histamine-induced H1-receptor internalisation”. Br. J. Pharmacol. 116 (6): 2715—23. PMC 1909113 Слободан приступ. PMID 8590995. 
  • Max SI, Chowdhury BA, Fraser CM (1996). „Sequence analysis of the 5'-untranslated region of the human H1 histamine receptor-encoding gene”. Gene. 171 (2): 309—10. PMID 8666296. doi:10.1016/0378-1119(96)00036-4. 
  • De Backer MD, Loonen I, Verhasselt P; et al. (1998). „Structure of the human histamine H1 receptor gene”. Biochem. J. 335 (3): 663—70. PMC 1219830 Слободан приступ. PMID 9794809. 
  • Horváth BV, Szalai C, Mándi Y; et al. (1999). „Histamine and histamine-receptor antagonists modify gene expression and biosynthesis of interferon gamma in peripheral human blood mononuclear cells and in CD19-depleted cell subsets”. Immunol. Lett. 70 (2): 95—9. PMID 10569698. doi:10.1016/S0165-2478(99)00126-1. 
  • Wang KY, Arima N, Higuchi S; et al. (2000). „Switch of histamine receptor expression from H2 to H1 during differentiation of monocytes into macrophages”. FEBS Lett. 473 (3): 345—8. PMID 10818238. doi:10.1016/S0014-5793(00)01560-X. 
  • Oda T, Morikawa N, Saito Y; et al. (2001). „Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes”. J. Biol. Chem. 275 (47): 36781—6. PMID 10973974. doi:10.1074/jbc.M006480200. 
  • Brew OB, Sullivan MH (2002). „Localisation of mRNAs for diamine oxidase and histamine receptors H1 and H2, at the feto-maternal interface of human pregnancy”. Inflamm. Res. 50 (9): 449—52. PMID 11603849. doi:10.1007/PL00000269. 
  • Gutzmer R, Langer K, Lisewski M; et al. (2002). „Expression and function of histamine receptors 1 and 2 on human monocyte-derived dendritic cells”. J. Allergy Clin. Immunol. 109 (3): 524—31. PMID 11898002. doi:10.1067/mai.2002.121944. 
  • Idzko M, la Sala A, Ferrari D; et al. (2002). „Expression and function of histamine receptors in human monocyte-derived dendritic cells”. J. Allergy Clin. Immunol. 109 (5): 839—46. PMID 11994709. doi:10.1067/mai.2002.124044. 

Vidi još

Преузето из „https://sr.wikipedia.org/w/index.php?title=Histaminski_H1_receptor&oldid=5522130”